I-Ticagrelor Newgreen Supply APIS 99% Ticagrelor Powder

Ukuchazwa Komkhiqizo
I-Ticagrelor iyimbangela ye-antipretlet, i-P2Y12 Receptor Antaing, esetshenziselwa ukuvikela izehlakalo zenhliziyo, ikakhulukazi ezigulini ezine-coronary syndrome (ACS). Yehlisa ubungozi be-thrombosis ngokuvimbela ukuhlanganiswa kwe-platelet.
Mechanics Main
Vimbela ukuhlanganiswa kwe-platelet:
I-Ticagrelor ibuyele emuva ku-P2Y12 receptor entweni yeplatelet, kuvimbela ukusebenza kwe-Platelet kanye nokuhlanganiswa okubangelwa yi-adenosine diphosphate (ADP), ngaleyo ndlela kunciphisa ukwakheka kwe-thrombus.
Izinkomba
I-Ticagrelor isetshenziswa ikakhulukazi kulezi zimo ezilandelayo:
I-Acute Coronary Syndrome:Kubandakanya iziguli ezine-angina ezingazinzile kanye ne-MyOCardial infarction, imvamisa esetshenziswa ngokuhlanganiswa ne-aspirin ukunciphisa ubungozi bezehlakalo zenhliziyo.
Ukuvimbela Kwesekondari Yezehlakalo Zezinhliziyo Zenhliziyo:Ezigulini ezivele zinomcimbi wenhliziyo ukuvimbela enye.
Coha
Into | Ukucacisa | Umphumela |
Ukubonakala | Umhlophe we-powder | Qhubelelayo |
Hlela | -Yisimilo | Qhubelelayo |
Ngalokho | ≥99.0% | 99.8% |
-Nembelelekile | -Yisimilo | Qhubelelayo |
Ukulahleka kokuwomile | 4-7 (%) | 4.12% |
Inani eliphelele | I-8% max | 4.85% |
Insimbi esindayo | ≤10 (PPM) | Qhubelelayo |
I-Arsenic (as) | 0.5ppm max | Qhubelelayo |
Ukuhola (PB) | 1ppm max | Qhubelelayo |
I-Mercury (HG) | I-0.1ppm max | Qhubelelayo |
Isibalo sepuleti esiphelele | I-10000cFu / g max. | I-100cFU / g |
I-Yeast & Mold | I-100cFU / g max. | >I-20cFU / g |
Salmonella | -Phikisayo | Qhubelelayo |
E.coli. | -Phikisayo | Qhubelelayo |
Staphylococcus | -Phikisayo | Qhubelelayo |
Ukugcina | -Nokwazi | |
Ukubeka | Gcina endaweni evaliwe kahle ngamazinga okushisa aphansi njalo futhi akukho ukukhanya kwelanga okuqondile. | |
Impilo yeshelufu | Iminyaka emi-2 lapho igcinwa kahle |
Umphumela wecala
I-Ticagrelor ngokuvamile ibekezelelwa kahle, kepha eminye imiphumela emibi kungenzeka, kufaka phakathi:
Isopha:Umphumela ojwayelekile ojwayelekile, ongaba nomphumela wezehlakalo ezithambile noma ezinzima zokopha.
Ubunzima bokuphefumula:Ezinye iziguli zingathola ubunzima bokuphefumula noma ukukhwehlela.
Ukusabela kwesisu:njenge-nausea, ubuhlungu besisu noma ukugayeka.
Amanothi
Ingozi yokuphamba:Ingozi yokopha kufanele ibhekwe njalo lapho usebenzisa iTicagrelor, ikakhulukazi lapho isetshenziswa ngokuhlangenwe nakho nezinye izidakamizwa eziphikisayo.
Umsebenzi we-Hepatic:Sebenzisa ngokuqapha ezigulini ezinokukhubazeka kwe-hepatic; Ukulungiswa kwethamo kungadingeka.
Ukusebenzisana kwezidakamizwa:I-Ticagrelor ingaxhumana nezinye izidakamizwa. Kufanele utshele udokotela wakho ngazo zonke izidakamizwa ozithathayo ngaphambi kokuyisebenzisa.
Iphakheji nokulethwa


