Terbinafine hydrochloride high purrocloride apiretity API izinto ezibonakalayo i-78628-80-5

Ukuchazwa Komkhiqizo
Terbinafine hydrochlorideIngabe umuthi we-antifungal usetshenziselwa ukwelapha izifo ezahlukahlukene. Imvamisa ngesimo samathebulethi noma okhilimu. I-Terbinafine Hydrochloride umuthi ophumelelayo we-antifungal esetshenziswa ukwelapha ukutheleleka okuthe xaxa fungal. Noma ngabe kukhulunywa ngonyawo lwe-athlete noma izifo ze-fungal, le misebenzi yokuvimbela ukuvimbela ukukhiqizwa kwe-ergrestel futhi inikezela ngezinketho zohlelo lokusebenza lwe-topical neyomlomo ukuze kube lula kanye nokusebenza ngempumelelo.
Coha
Into | -Vamile | Umphumela wokuhlola |
Ngalokho | 99% | Kuvumelana |
Umbala | Umhlophe we-powder | Kuvumelana |
Iphunga | Alikho iphunga elikhethekile | Kuvumelana |
Usayizi wezinhlayiyana | I-100% idlula 80mesh | Kuvumelana |
Ukulahleka kokuwomile | ≤5.0% | I-2.35% |
Okuhlangene | ≤1.0% | Kuvumelana |
Insimbi esindayo | ≤10.0ppm | I-7ppm |
As | ≤2.0PPM | Kuvumelana |
Pb | ≤2.0PPM | Kuvumelana |
Izinsalela zokubulala izinambuzane | -Phikisayo | -Phikisayo |
Isibalo sepuleti esiphelele | ≤100cFU / g | Kuvumelana |
I-Yeast & Mold | ≤100cFU / g | Kuvumelana |
E.coli | -Phikisayo | -Phikisayo |
Salmonella | -Phikisayo | -Phikisayo |
Ukugcina | Xoxa ngokucaciswa | |
Ukubeka | Egcinwe endaweni epholile neyomile, gcina kude nokukhanya okuqinile nokushisa | |
Impilo yeshelufu | Iminyaka emi-2 lapho igcinwa kahle |
Sebenza
1.Terbinafine hydrochloride a anlyla antifungagal. Kuyinto ye-lipophilic kakhulu emvelweni futhi ivame ukuqongelela esikhunjeni, izipikili, nezicubu ezinamafutha.
I-2.interbinafine · HL Ilungu le-Allyl Class of Antifungela, litholakale liyi-inhibitor ethize ye-ergostel syntherthesis nge-squalene epoxidaseving. I-squalene epoxidase iyinzyme isikhunti dermatophyte ukudiliza i-squalene, ephazamisa umsebenzi we-membrane cell membrane kanye nokuhlanganiswa kodonga.
I-3.Interbinafine hydrochloride inomphumela we-fungicidal kwi-FungiDidal yesikhumba kanye nomphumela wokuvinjwa kuma-albician we-candida. Ilungele ukutheleleka kwesikhumba kanye nezipikili ezibangelwa yisikhunta esingesikhulu, njenge-ringworm, i-ringworm yomzimba, i-ringworm yezipikili, i-ringworm yezipikili i-rubrum ebangelwa i-trichophyton rubrum, i-microsporum canis kanye ne-flocculus epidermidis.
Isicelo
I-Terbinafine Hydrochloride iyimpuphu emhlophe enhle ye-crystalline powder ethambile ngokukhululekile ku-methan nase-dichlorome, incanel e-ethanol, futhi incane kancane emanzini. Njengamanye ama-allylamine, i-Terbinafine ivimbela ukuhlanganiswa kwe-ergorel ngokuvimbela i-squalene epoxidase,
I-enzyme eyingxenye ye-fungal cell membrane symbrane payway. Ngoba uTerbinafine uvimbela ukuguqulwa kweStsqualene kuya eLanosterol, i-ergorel ayikwazi ukuguqulwa. Lokhu kucatshangelwa ukuthi kushintsha ukufezekiswa kweseli ngokufanele, kubangele ukugcwala kwe-fungal cell.
1. I-Herbinafine Hcl iyasebenza kakhulu eqenjini le-Dermatophyte lesikhunta.
2. Njengo-1% ukhilimu noma i-powder, isetshenziswa kakhulu ekuthelelekeni kwesikhumba okuvela phezulu njenge-jock itch (tin cruris),
Unyawo lwe-Athlete (i-Tinea Pedis), nezinye izinhlobo ze-ringworm (i-tin Corpor ris). I-Terbinafine Cream isebenza cishe ngesigamu sesikhathi esidingekayo
ngamanye ama-antifungela.
3. I-ORAL 250MG amatafula avame ukubekelwa ukwelashwa kwe-Onychomycosis, ukutheleleka nge-fungal nail, ngokuvamile yi-dermatophyte
noma izinhlobo ze-candida. Ukutheleleka kwezikhunta ze-fungal zitholakala ekujuleni ngaphansi kwesipikili ku-cuticle lapho kusetshenziswe khona izindlela zokwelapha eziphezulu
abakwazi ukungena ngamanani anele. Izibhebhe zingahle, kuyaqabukela, zibangele i-hepatotoxicity, ngakho-ke iziguli zixwayiswa ngalokhu futhi
ingahle ibhekwe ngezivivinyo zokusebenza kwesibindi. Ezinye izindlela zokuphatha ngomlomo zifundelwe.
I-4. I-Terbinafine ingahle incishise noma ikhulise amandla ama-supus cuteous lupus erythematosus. Abantu abane-lupus erythematosus kufanele
Okokuqala xoxa ngezingozi ezingaba khona nodokotela wazo ngaphambi kokuqalwa kokwelashwa.
Imikhiqizo ehlobene
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