I-Terbinafine HydrochloriderIka i-Pulty Api pulty Api Prospas 78628-80-50-5

Ingcaciso yeMveliso
I-terbinafine hydrochlorideNgaba amayeza e-antifungal asetyenziselwa ukuphatha ngeendlela ezahlukeneyo. Ngokwesiqhelo ngohlobo lweetafile okanye iikhrim. I-Terbinafine Hydrochloride i-rolldrochloride yenziwa ngamayeza asebenzayo asebenzayo okunyanga usulelo oluninzi lwefungi. Nokuba kujongana nolusu lwe-Itleete okanye usulelo lwe-fungal, le ndlu ye-fungal, le nkqubo ye-Ergosterol imveliso kwaye ibonelela ngeendlela eziphezulu kunye nempumelelo.
Coa
Izinto | Umgangatho | Iziphumo zovavanyo |
I-assay | I-99% | Ivumelana |
Umbala | Umgubo omhlophe | Ivumelana |
Ivumba | Akukho phunga likhethekileyo | Ivumelana |
Ubungakanani bentsundu | I-100% ye-80mesh | Ivumelana |
Ilahleko yokomisa | ≤5.0% | I-2.35% |
Intsalela | ≤1.0% | Ivumelana |
Intsimbi enzima | ≤10.0ppm | I-7ppm |
As | ≤2.0ppm | Ivumelana |
Pb | ≤2.0ppm | Ivumelana |
Intsalela yamayeza | Engalunganga | Engalunganga |
I-pile itreyini | ≤100cfu / g | Ivumelana |
I-Youst & Ibumba | ≤100cfu / g | Ivumelana |
E.coli | Engalunganga | Engalunganga |
Isalmonella | Engalunganga | Engalunganga |
Ukuqukumbela | Ivumelana nenkcazo | |
Ukugcinwa | Igcinwe kwindawo epholileyo neyomileyo, gcina kude kukhanyiso nobutshinga | |
Beka ubomi kwishelufa | Iminyaka emi-2 xa igcinwe ngokufanelekileyo |
Umsebenzi
I-1.Terbhinafine Hydrochloride i-allyla antifungal. Yi-lipiflic kakhulu kwindalo kwaye idla ngokuqokelela kwisikhumba, izikhonkwane, kunye nezicubu ezinamafutha.
I-2.mterbinafinefine · · hcl yeklasi ye-Allyl ye-antifosteals, ifunyenwe ingu-Ergosterol Synthesis nge-squalese epoxidase. I-squalene Epoxidase yi-enzyme ikhutshwe yi-Dermatophyte Fungi ukuze iphule i-squalene, eyaphazamisa umsebenzi we-membrane yeseli kunye noWall Synthesis.
I-3.2 i-Herterbifafine hydrochloride inefuthe le-funglical kwi-fungi kunye nefuthe le-Albicans. Ilungele ulusu kunye nosulelo lwezipikili obangelwa yi-fungficialial fungficial, iringi ye-ringworm ye-femur, iringworm ye-biricar, i-ringworm ye-iriclum rubrum ye-Triaphyton ye-Tridermidis.
Isicelo
I-Terbinafine Hydrochloride yi-crystalline ye-crystalline ye-crystalline ye-crystalline enyibilikisi e-methan naseDichlorome, inyibilikiswe e-ethanol, kwaye inyibilikiswe e-ethanol, kwaye inyibilikiswe e-ethanol, kwaye inyibilike inyibilikisi emanzini. Njengaye amanye iAllylamines, i-terbinafine ithintela i-Ergosterol Synthesis ngu-ethintela i-squalese,
I-enzyme enenxalenye ye-fungrane selm ye-fungline syntheaway. Kungenxa yokuba i-terbinafine ithintela i-ofisi yoguquguquko kwi-lanosterol, i-ergosterol ayinakudityaniswa. Oku kucingelwa ukutshintsha i-membrane yeseli, kubangela i-lysis ye-funglicy.
I-1. I-TerbinaFine HCL ikakhulu isebenza ikakhulu kwiqela le-dermatophyte yefungi.
2. Njenge-Cream eyi-1% okanye i-powder, isetyenziswa ngokugqibeleleyo kusulelo olugqibeleleyo lolusu olunjenge-jock itch (iTinea cruris),
Unyawo lweembaleki (i-tinea pedis), kunye nezinye iintlobo ze-ringworm (i-tinea boris). I-Terbinafine Cream isebenza malunga nesiqingatha sexesha elifunekayo
ngolunye uhlobo.
I-3. Iitafile ze-250mg ezingama-250mg zihlala zimiselwa kunyango lwe-onychomycosis, i-fungal yosulelo, ngokwesiqhelo yi-dermatophyte
okanye iintlobo zeNtu. Usulelo lwezipikili zefunga lubekwe ngaphakathi kwephayini kwi-cutecle apho unyango olusetyenzisiweyo
abakwazi ukungena ngexabiso elaneleyo. Amacwecwe anokuthi, kunqabile, ukubangela i-hepatocity, ke abaguli balumkisiwe ngale nto kwaye
inokubekwa esweni kunye neemvavanyo zomsebenzi weSibindi. Iindlela ezizezinye kulawulo ngomlomo zifundiwe.
I-4. I-Terbinafine inokuphelisa okanye ivusele i-lupus ye-suremane ye-cythemaotos. Abantu abanee-lupus erythematosis kufuneka
Okokuqala Xoxa ngengozi kugqirha wabo ngaphambi kokuqalisa unyango.
Iimveliso ezinxulumene noko
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