Terbinafine hydrochloride dị elu dị elu API ihe onwunwe nke 78628-80-5

Nkọwa nke ngwaahịa
Terbinafine hydrochloridebụ ọgwụ antifung na-emeso ọtụtụ ọrịa dị iche iche. Ọ na-abụkarị n'ụdị mbadamba ma ọ bụ ude. Terbinafine hydrochloride bụ ọgwụ antifungal dị irè iji gwọọ ọrịa dị iche iche fungal dị iche iche. Ma ọ na-agwa ya okwu na-efe efe ma ọ bụ fungal ntu, ọrụ ọgwụ a site na-egbochi mmepụta ergobel ma na-enye ma ngwa ọrụ maka ịdị mma na ịdị irè.
Iko
Ihe | Standadi | Nsonaazụ nnwale |
Nke oma | 99% | Kwekọrọ |
Agba | Ntụ ntụ | Kwekọrọ |
Isi | Ọ dịghị isi na-acha uhie uhie | Kwekọrọ |
Urughuru | 100% Pass 80mesh | Kwekọrọ |
Mfu na ihicha | ≤5.0% | 2.35% |
Yedue | ≤1.0% | Kwekọrọ |
Ígwè oke | ≤10.0ppm | 7ppm |
As | ≤2.0ppm | Kwekọrọ |
Pb | ≤2.0ppm | Kwekọrọ |
Ọgbụgba na-egbu egbu | Nju | Nju |
Mkpokọta ọnụ ọgụgụ | ≤100cU / g | Kwekọrọ |
Yist & Ebu | ≤100cU / g | Kwekọrọ |
Exlili | Nju | Nju |
Salmonella | Nju | Nju |
Mmechi | Njikọ na nkọwapụta | |
Storaji | Echekwara na Cool & Akọrọ, na-ahapụ ìhè na okpomoku | |
Ndụ Ndụ | Afọ 2 mgbe echekwara nke ọma |
Oru oruru
1.Tterbinafine hydrochloride a Allyla antifungal. Ọ bụ oke lopophilic na okike ma na-enwekwa ihe na-agbakọta anụ ahụ, mbọ, na anụ ahụ abụba.
2.Trbinafine hlr so na klas Antifunsicals, ahụla ka ọ bụrụ otu onye na-egbochi nje na-egbochi ọrịa ergobel site na mgbochi epoxdase. Squalene epoxdase bụ enzyme wepụtara site na Dermatophypyte fungi iji mebie squalene, nke na-egbochi ya na ọrụ akpụkpọ ụkwụ na mgbidi.
3.tersbinafine hydrochloride nwere mmetụta na-atọ ụtọ na akpụkpọ ahụ na-egbu egbu na mmetụta na-egbochi infida Albicans. Ọ dị mma maka anụ ahụ na ntu na-enweghị atụ nke fungim nke anụ ahụ, na-anyụkwa akwara nke anụ ahụ, microsporum Canis na Flosculus Epidermidis kpatara.
Akwukwo icho oru
Terbinafine hydrochloride bụ ezigbo kristal ntụ ntụ nke na-acha ọcha nke na-acha na methan na Dichlorome, soluble na ethanol, ma dịtụ na mmiri. Dị ka allinlanines ndị ọzọ, Tarbinafine na-egbochi njigide ngwa ngwa site na igbochi squalene epoxdase,
Otu enzyme nke bụ akụkụ nke fungane sel membrane sysis. N'ihi na terbinafine na-egbochi ntụgharị nke Lanorol, ergorol enweghị ike ịhazi. A na-eche na ị gbanwee ihe omume nke celmmbrane permeability, na-akpata fungal cell lysis.
1
2. Dị ka 1% ude ma ọ bụ ntụ ntụ, a na-eji ya eme ihe maka ọrịa anụ ahụ dị ka JCOCET),
Twokwụ nke egwuregwu (Tinia Pedis), na ụdị mgbaaka ndị ọzọ (Tinea Corpors). Terbinafine na-eto eto na-arụ ọrụ na ọkara oge achọrọ
site na antifunges ndị ọzọ.
3. A na-etinyekarị mbadamba 250mgs 250mg maka ọgwụgwọ Onchemiscosis, ọrịa ụynal, na-abụkarị site na dermatophyte
ma ọ bụ ụdị nkà. Ọrịa ntu na-efe efe dị omimi n'okpuru ntu na okirikiri nke ọgwụgwọ etinyere
enweghị ike ịbanye na oke zuru ezu. Mbadamba nkume ahụ nwere ike, adịkarịghị, na-akpata Hepatotoxicity, yabụ a dọrọ ndị ọrịa aka na ntị nke a
enwere ike inyocha ule imeju. Ndị ọzọ amụrụla nchịkwa.
4. Trubinafine nwere ike ịmegharị ma ọ bụ na-ewe iwe na substactute sublatactute ntakịrị lepus erythematosus. Ndị nwere lyupus erythematosus kwesịrị
Buru ụzọ tụrịta ihe egwu ndị dọkịta ha nwere tupu ịmalite ọgwụgwọ.
Ngwaahịa metụtara
Newlọ ọrụ mmepụta ọhụụ na-enyekwa Amino acid dị ka ndị na-eso:

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