Ihe ngosi ohuru ohuru nke Ibudilast di elu 99% ibudulast ntụ ntụ

Nkọwa nke ngwaahịa
Ibubilast bụ ọgwụ nke a na-eji eme ihe ọtụtụ ọrịa akwara ozi na ọrịa inflayrated. Ihe ndị a bụ mmeghe nke echiche:
Ọrịa akwara ozi: Ibudilast egosila uru enwere ike ịba uru na ụfọdụ ọmụmụ maka ọtụtụ sclerosis (ms), ọrịa Alzheimer, na ọrịa akwara ọzọ.
Nchịkwa mgbu: A na-ejikwa ya eme ihe mgbu na-adịghị ala ala, ọkachasị mgbe metụtara ihe mgbu na neuropaatheric.
Asthma na nsogbu nfụka: A na-ejikwa Ibudilast n'ihe ụfọdụ iji gwọọ ashie na nsogbu nfụkasị.
Oganihu
Ibubilast egosila ikike ịrụ ọrụ na ụfọdụ ọrịa akwara ozi na ọnwụnwa na-arụsi ọrụ ike, ọkachasị na ịkagbu ọrịa na-adịghị mma ma melite mgbaàmà. Agbanyeghị, ọ dị mkpa nyocha ọzọ iji kwado nsonaazụ ya ogologo na nchekwa.
Na mmechi, ibubilast bụ ọgwụ nwere ike iji ọtụtụ ngwa, na-ekwe nkwa na ọgwụgwọ nke nsogbu akwara na ọrịa inflocalted. Ekwesịrị iji ya mee ihe n'okpuru nduzi nke dibịa ma nyochaa ya mgbe niile.
Iko
Asambodo Nnyocha
Ihe | Nkowa | Nsonaazụ |
Mputa | Ruthite ma ọ bụ ntụ ntụ | Ntụ ntụ |
Nchọpụta HPLC | Kwekọrọ na ntụnye aka Oge nnabata kachasị elu | Kwekọrọ |
Ntugharị kpọnwụrụ iche | + 20.0. + 22.0. | +1. |
Ochie ọla dị arọ | ≤ 10pm | <10ppm |
PH | 7.58.5 | 8.-8 |
Mfu na ihicha | ≤ 1.0% | 0.25% |
Izizi | ≤3ppm | Kwekọrọ |
Arsenic | ≤1pm | Kwekọrọ |
Kengwe | ≤1pm | Kwekọrọ |
Merlury | ≤0. 1ppm | Kwekọrọ |
Na-agbaze | 250.0℃~ 265.0℃ | 254.7 ~ 255.8℃ |
Tọgharịa na mgbanye | ≤0. 1% | 0.03% |
Hydrazine | ≤2ppm | Kwekọrọ |
Nnukwu njupụta | / | 0.21G / ml |
Nnọọ njupụta | / | 0.45g / ml |
Asambodo (Ibubiast) | 99.0% ~ 101.0% | 99.65% |
Ngụkọta Aerobes | ≤1000cfu / g | <2cfu / g |
Ebu & yists | ≤100cU / g | <2cfu / g |
Exlili | Nju | Nju |
Salmonella | Nju | Nju |
Storaji | Chekwaa na ebe dị jụụ & ihicha, na-eme ka ìhè siri ike. | |
Mmechi | Tozuru oke |
Oru oruru
Ibubilast bụ ọgwụ a na-eji emeso ọtụtụ ọrịa akwara ozi. Ọrụ ya gụnyere:
1. Antiinflamtory mmetụta:Ibubilast nwere ihe mgbochi na-emegide ya ma nwee ike igbochi mmeghachi omume na sistemụ akwara, nke na-eme ka ọ dị na ọgwụgwọ ọrịa akwara metụtara na mbufụt.
2. Neuroprotoctions:Ekwenyere na Ibudilast nwere mmetụta na-emetụta ihe na-eme, ikekwe na-echebe usoro ụjọ site na ibelata ihe na-emebi akwara ọbara na ọnwụ.
3. Ndị na-eme ka ọrụ akwara ozi:N'ebe ụfọdụ ọmụmụ, Ibubiastis egosila ike iji meziwanye ọrụ akwara, karịsịa na ndị ọrịa nwere ọtụtụ sclerosis (ms) na ọrịa neurodegenerited.
4. Na-egbochi mwepụta nke neurotronsmitters:Ibubilast nwere ike rụọ ọrụ site na idozi mwepụta nke neurotronsmitters, na-emetụta nnyefe nke akara akwara.
5. Maka njikwa ihe mgbu:A mụworị Ibudilast maka njikwa nke na-adịghị ala ala n'ọnọdụ ụfọdụ, ọkachasị mgbe metụtara ihe mgbu neuropatheric.
Na mmechi, Ibubilast bụ ọgwụ na ọtụtụ nsonaazụ, nke eji eji ọgwụgwọ ọrịa akwara ọrịa, karịsịa na mpaghara nke mbufụt na neuroprotoctions. Ekwesịrị iji ya mee ihe n'okpuru nduzi nke dibịa ma nyochaa ya na onye ikpe.
Akwukwo icho oru
Ngwa nke ibudilast na-eme nke ọma n'akụkụ ndị a:
1. Ọrịa ụjọ na-atụ ụjọ:
Otutu sclerosis (ms): ibudilast na-egosi ike arụmọrụ arụmọrụ na ọgwụgwọ nke ọtụtụ sclerosis ma nwee ike inyere gị aka na ọrịa ọ bụla ma melite mgbaàmà.
Ọrịa Alzheimer: ụfọdụ ọmụmụ egosila na Ibubiastilast nwere ike meziwanye ọrụ ndị ọrịa na ọrịa Alzheimer.
2. Nchịkwa mgbu:
Nuuropatheric mgbu: A na-amụ Ibudilast maka ọgwụgwọ nke ihe mgbu na-adịghị ala ala jikọtara mmebi akwara, dịka shuga diopathy na posthetic na ọkwa na ọkwa.
3. Ọrịa iku ume:
Asthma na nsogbu nfụkasị: A na-eji mBudilast n'ụzọ ụfọdụ iji gwọọ asthma na nsogbu nfụkasị ya nwere ike inye aka belata mgbaàmà.
4. Mpaghara nyocha ndị ọzọ:
A na-enyocha Mybudilast n'oge ọnwụnwa maka nsogbu ndị ọzọ na ọnọdụ ahụike, dịka ịda mba na nchegbu.
Na nchịkọta, Ibubilast nwere ọtụtụ ngwa, na-elekwasị anya na ọgwụgwọ ọrịa akwara, njikwa mgbu, yana ụfọdụ ọrịa iku ume. N'agbanyeghị nnukwu ọrụ ya, ọ dị mkpa ịgbaso nduzi dọkịta mgbe ị na-eji ya ma na-elebara ọganihu nke nyocha nke ụlọ ọgwụ dị mkpa.
Ihe ngwugwu & nnyefe


